Compile Data Set for Download or QSAR
Found 9 of ic50 data for polymerid = 50003871
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.469nMAssay Description:Inhibition of human TAOK1 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human TAOK1 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50429615(CHEMBL2334586)copy SMILEScopy InChI
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP5771PubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50329427(5-(2-Amino-pyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-c...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of TAO1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6JM3PubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50507430(CHEMBL3937369)copy SMILEScopy InChI
Affinity DataIC50: 490nMAssay Description:Inhibition recombinant human TAOK1 (1 to 356 residues) after 5 mins in presence of [33P] ATP by Topcount methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ7214PubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50429867(CHEMBL2333365)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TAO1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC847XPubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human TAO1 (1 to 327 residues) using myelin basic protein as substrate incubated for 40 mins in presence of [gamma33P]ATP b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TAOK1 using MBP substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetSerine/threonine-protein kinase TAO1(Homo sapiens (Human))TBA
LigandPNGBDBM50401152(CHEMBL2205766)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TAOK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ412BPubMed